SCHEMBL20002176

SCHEMBL20002176

N#CC1(C(=O)N2CCC([S+]([O-])c3ccc(F)cc3)C2)CCNCC1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 3/20 0.38
RORC P51449 4/20 0.37
JAK1 P23458 1/20 0.33
JAK3 P52333 1/20 0.33
CNR2 P34972 1/20 0.33
HSD11B1 P28845 6/20 0.32
DPP4 P27487 1/20 0.32
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
ATM Q13315 1/20 0.31
CTSB P07858 1/20 0.31
CTSS P25774 1/20 0.31
CTSK P43235 1/20 0.31
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002166 0.82 RORC (0.40) TACR3RORCCNR2HSD11B1DPP4
SCHEMBL20003044 0.76 RORC (0.40) RORCNPC1RAB9AATM
SCHEMBL20003139 0.74 RAB9A (0.33) RORCHSD11B1DPP4NPC1RAB9A
SCHEMBL20002445 0.74 RORC (0.41) RORCHSD11B1NPC1RAB9AATM
SCHEMBL20002171 0.74 KMT2A (0.38) RORCHSD11B1NPC1RAB9AATM
SCHEMBL20003241 0.74 RORC (0.41) RORCHSD11B1NPC1RAB9AATM
SCHEMBL20002856 0.74 RORC (0.42) RORCHSD11B1DPP4NPC1RAB9A
SCHEMBL20002926 0.74 RORC (0.43) RORCDPP4KCNH2
SCHEMBL20002207 0.74 RORC (0.45) RORCNPC1RAB9AATM
SCHEMBL20002924 0.73 MAPK1 (0.34) RORCHSD11B1NPC1RAB9AATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed