SCHEMBL20003139

SCHEMBL20003139

O=C(N1CCC([S+]([O-])c2ccc(F)cc2)C1)C1(F)CCSCC1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.33
NPC1 O15118 2/20 0.33
ATM Q13315 1/20 0.33
NR1I2 O75469 1/20 0.33
RORC P51449 1/20 0.33
CYP2C19 P33261 1/20 0.32
EPHX2 P34913 1/20 0.32
HSD11B1 P28845 7/20 0.32
MMP1 P03956 1/20 0.31
MMP13 P45452 1/20 0.31
DPP4 P27487 1/20 0.31
DPP8 Q6V1X1 1/20 0.31
DPP9 Q86TI2 1/20 0.31
MAPK1 P28482 1/20 0.31
MAPT P10636 3/20 0.31
HRH3 Q9Y5N1 1/20 0.30
PARP10 Q53GL7 1/20 0.30
LMNA P02545 1/20 0.30
KMT2A Q03164 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20003092 0.85 RORC (0.33) RAB9ANPC1ATMRORCMAPK1
SCHEMBL20003044 0.80 RORC (0.40) RAB9ANPC1ATMRORCMAPT
SCHEMBL20002445 0.78 RORC (0.41) RAB9ANPC1ATMRORCHSD11B1
SCHEMBL20002171 0.78 KMT2A (0.38) RAB9ANPC1ATMRORCHSD11B1
SCHEMBL20003241 0.78 RORC (0.41) RAB9ANPC1ATMRORCHSD11B1
SCHEMBL20002926 0.77 RORC (0.43) NR1I2RORCDPP4MAPK1
SCHEMBL20002856 0.77 RORC (0.42) RAB9ANPC1ATMRORCHSD11B1
SCHEMBL20002207 0.77 RORC (0.45) RAB9ANPC1ATMNR1I2RORC
SCHEMBL20003052 0.76 HSD11B1 (0.38) RAB9ANPC1ATMNR1I2RORC
SCHEMBL20002748 0.76 RORC (0.39) RAB9ANPC1ATMRORCHSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed