SCHEMBL20002230

SCHEMBL20002230

CCc1cc([S+]([O-])C2CCN(C(=O)C3CCCCC3)C2)ccc1F

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MTNR1B P49286 1/20 0.41
HSD11B1 P28845 2/20 0.39
GAA P10253 1/20 0.38
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
ALDH1A1 P00352 4/20 0.36
RORC P51449 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
TACR3 P29371 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002759 0.85 GFER (0.43) HSD11B1GAAMEN1KMT2AALDH1A1
SCHEMBL20002698 0.82 HSD11B1 (0.47) HSD11B1MEN1KMT2AALDH1A1RORC
SCHEMBL20002706 0.82 HSD11B1 (0.47) HSD11B1MEN1KMT2AALDH1A1RORC
SCHEMBL20002995 0.81 GFER (0.50) HSD11B1MEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL20002574 0.80 ALDH1A1 (0.51) MEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL20002641 0.79 TDP1 (0.42) HSD11B1MEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL20003010 0.78 RORC (0.43) MTNR1BALDH1A1RORC
SCHEMBL20003089 0.78 GPR183 (0.45) HSD11B1MEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL20002705 0.78 ALDH1A1 (0.41) HSD11B1MEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL20002746 0.77 CCR5 (0.44) HSD11B1MEN1KMT2AALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed