SCHEMBL20003089

SCHEMBL20003089

O=C(C1CCCCC1)N1CCC([S+]([O-])c2ccc(Br)cc2)C1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GPR183 P32249 1/20 0.45
KMT2A Q03164 3/20 0.42
MEN1 O00255 2/20 0.42
GHSR Q92847 1/20 0.41
ALDH1A1 P00352 2/20 0.41
TSHR P16473 1/20 0.41
EPHX2 P34913 1/20 0.39
MMP1 P03956 1/20 0.39
MMP3 P08254 1/20 0.39
MMP7 P09237 1/20 0.39
MMP9 P14780 1/20 0.39
MMP13 P45452 1/20 0.39
PTPN1 P18031 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
KEAP1 Q14145 1/20 0.39
RXFP1 Q9HBX9 1/20 0.38
HSD11B1 P28845 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
CCR5 P51681 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002641 0.89 TDP1 (0.42) KMT2AMEN1ALDH1A1TSHRMMP1
SCHEMBL20002705 0.88 ALDH1A1 (0.41) KMT2AMEN1ALDH1A1TSHRMMP1
SCHEMBL20002706 0.88 HSD11B1 (0.47) KMT2AMEN1ALDH1A1TSHREPHX2
SCHEMBL20002574 0.88 ALDH1A1 (0.51) KMT2AMEN1ALDH1A1TSHREPHX2
SCHEMBL20002698 0.88 HSD11B1 (0.47) KMT2AMEN1ALDH1A1TSHREPHX2
SCHEMBL20002746 0.86 CCR5 (0.44) KMT2AMEN1ALDH1A1TSHRPTPN1
SCHEMBL20002660 0.85 FASN (0.52) KMT2AMEN1GHSRTSHRPTPN1
SCHEMBL20003098 0.84 GPR183 (0.38) GPR183KMT2AMEN1ALDH1A1TSHR
SCHEMBL20002932 0.84 KDM1A (0.42) KMT2AMEN1ALDH1A1TSHREPHX2
SCHEMBL20002995 0.82 GFER (0.50) KMT2AMEN1ALDH1A1TSHRMMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed