SCHEMBL20002352

SCHEMBL20002352

C[S+]([O-])NC(=O)C1CCN(C(=O)N2CCC([S+]([O-])c3ccc(F)cc3)C2)CC1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.39
EPHX2 P34913 1/20 0.37
PTPN1 P18031 1/20 0.37
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
POLB P06746 1/20 0.36
LMNA P02545 3/20 0.36
ALDH1A1 P00352 2/20 0.36
TSHR P16473 1/20 0.36
HTT P42858 1/20 0.36
PKM P14618 1/20 0.36
HSD11B1 P28845 3/20 0.35
RORC P51449 1/20 0.35
KMT2A Q03164 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
UBE2M P61081 1/20 0.35
DCUN1D1 Q96GG9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002669 0.84 NOTUM (0.45) MAPTLMNAALDH1A1HSD11B1RORC
SCHEMBL20002969 0.84 NOTUM (0.45) MAPTLMNAALDH1A1HSD11B1RORC
SCHEMBL20002964 0.84 RORC (0.35) EPHX2HDAC3HDAC1HDAC2RORC
SCHEMBL20002280 0.82 TACR1 (0.40) HDAC3HDAC1HDAC2PKMHSD11B1
SCHEMBL20002958 0.82 NOTUM (0.48) MAPTEPHX2POLBLMNAALDH1A1
SCHEMBL20002957 0.82 NOTUM (0.48) MAPTEPHX2POLBLMNAALDH1A1
SCHEMBL20002167 0.82 KDM1A (0.40) EPHX2LMNAALDH1A1HTTPKM
SCHEMBL20003029 0.81 RORC (0.41) RORC
SCHEMBL20003049 0.80 AKR1C3 (0.51) EPHX2LMNAALDH1A1HTTPKM
SCHEMBL20003037 0.79 RORC (0.38) MAPTHDAC3HDAC1HDAC2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed