SCHEMBL20002964

SCHEMBL20002964

C[S+]([O-])NC1(C)CCN(C(=O)N2CCC([S+]([O-])c3ccc(F)cc3)C2)CC1

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
RORC P51449 7/20 0.35
GFER P55789 1/20 0.34
MCHR1 Q99705 1/20 0.34
KDM1A O60341 3/20 0.32
KMT2A Q03164 1/20 0.32
HDAC3 O15379 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC2 Q92769 1/20 0.32
EPHX2 P34913 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20003037 0.89 RORC (0.38) RORCGFERHDAC3HDAC1HDAC2
SCHEMBL20003029 0.87 RORC (0.41) RORCKDM1A
SCHEMBL20002352 0.84 MAPT (0.39) RORCKMT2AHDAC3HDAC1HDAC2
SCHEMBL20002167 0.81 KDM1A (0.40) RORCKDM1AEPHX2
SCHEMBL20002280 0.81 TACR1 (0.40) RORCHDAC3HDAC1HDAC2
SCHEMBL20002969 0.79 NOTUM (0.45) RORCKMT2A
SCHEMBL20003049 0.79 AKR1C3 (0.51) KMT2AEPHX2CYP2C19
SCHEMBL20002669 0.79 NOTUM (0.45) RORCKMT2A
SCHEMBL20002631 0.78 HSD11B1 (0.33) RORCKMT2A
SCHEMBL20002664 0.78 TSHR (0.41) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed