SCHEMBL20002813

SCHEMBL20002813

CC(OCc1ccc(F)cc1F)(C(F)(F)F)C(F)(F)F

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 5/20 0.53
AGXT P21549 2/20 0.53
MAOB P27338 1/20 0.43
RORC P51449 2/20 0.41
RIPK1 Q13546 2/20 0.39
GSK3B P49841 1/20 0.37
BACE1 P56817 1/20 0.37
KDM4E B2RXH2 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
TRPA1 O75762 1/20 0.35
MAPK14 Q16539 2/20 0.35
HTR6 P50406 1/20 0.34
NR3C1 P04150 1/20 0.34
PGR P06401 1/20 0.34
NR3C2 P08235 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002817 0.86 RORC (0.41) IDO1AGXTRORCRIPK1NR3C1
SCHEMBL16886252 0.85 IDO1 (0.51) IDO1AGXTMAOBRORCRIPK1
SCHEMBL13882408 0.84 IDO1 (0.58) IDO1AGXTMAOBRORCRIPK1
SCHEMBL20002764 0.80 NR3C1 (0.46) IDO1RORCMAPK14NR3C1PGR
SCHEMBL20002788 0.77 RORC (0.36) RORCRIPK1
SCHEMBL10202639 0.74 IDO1 (0.55) IDO1AGXTMAOBRIPK1GSK3B
SCHEMBL706473 0.74 IDO1 (0.64) IDO1AGXTMAOBRIPK1GSK3B
SCHEMBL16886255 0.73 IDO1 (0.41) IDO1AGXTRORCRIPK1NR3C1
SCHEMBL29467207 0.73 IDO1 (0.69) IDO1AGXTMAOBGSK3BBACE1
SCHEMBL27106193 0.71 IDO1 (0.56) IDO1AGXTMAOBRIPK1GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed