SCHEMBL20002817

SCHEMBL20002817

CC(OCc1cc(F)ccc1F)(C(F)(F)F)C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORC P51449 3/20 0.41
HTR2C P28335 5/20 0.41
SLC6A4 P31645 5/20 0.41
HTR2A P28223 4/20 0.40
RIPK1 Q13546 1/20 0.40
IDO1 P14902 5/20 0.39
NR3C2 P08235 2/20 0.39
NR3C1 P04150 1/20 0.39
CACNA1C Q13936 1/20 0.37
AGXT P21549 2/20 0.37
MMP2 P08253 2/20 0.37
MMP12 P39900 2/20 0.37
MMP1 P03956 1/20 0.37
MMP9 P14780 1/20 0.37
CA3 P07451 1/20 0.35
CA6 P23280 1/20 0.35
CA5A P35218 1/20 0.35
CA9 Q16790 1/20 0.35
CA14 Q9ULX7 1/20 0.35
CA5B Q9Y2D0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002813 0.86 IDO1 (0.53) RORCRIPK1IDO1NR3C2NR3C1
SCHEMBL18213802 0.84 HTR2C (0.43) RORCHTR2CSLC6A4HTR2ARIPK1
SCHEMBL16886255 0.83 IDO1 (0.41) RORCHTR2CSLC6A4HTR2ARIPK1
SCHEMBL12016019 0.74 IDO1 (0.44) HTR2CSLC6A4HTR2ARIPK1IDO1
SCHEMBL20002788 0.73 RORC (0.36) RORCRIPK1MMP2MMP12MMP1
SCHEMBL16886252 0.71 IDO1 (0.51) RORCRIPK1IDO1NR3C2NR3C1
SCHEMBL20002764 0.70 NR3C1 (0.46) RORCIDO1NR3C2NR3C1
SCHEMBL14763555 0.70 CACNA1C (0.50) HTR2CSLC6A4HTR2ARIPK1IDO1
SCHEMBL17217576 0.70 HTR2C (0.40) HTR2CSLC6A4HTR2ARIPK1IDO1
SCHEMBL13544214 0.70 MMP2 (0.50) HTR2CSLC6A4HTR2ARIPK1MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed