SCHEMBL20002932

SCHEMBL20002932

N#Cc1ccc([S+]([O-])C2CCN(C(=O)C3CCCCC3)C2)cc1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 4/20 0.42
EPHX2 P34913 2/20 0.42
MEN1 O00255 3/20 0.41
PAX8 Q06710 1/20 0.41
KCNH2 Q12809 1/20 0.40
KCNK3 O14649 2/20 0.39
KCNK9 Q9NPC2 2/20 0.39
ATM Q13315 1/20 0.39
FASN P49327 1/20 0.39
PRKAA2 P54646 1/20 0.38
ALDH1A1 P00352 1/20 0.38
TSHR P16473 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
KMT2A Q03164 2/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
PTPN1 P18031 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002641 0.85 TDP1 (0.42) MEN1ALDH1A1TSHRKMT2APTPN1
SCHEMBL20003089 0.84 GPR183 (0.45) EPHX2MEN1ALDH1A1TSHRKMT2A
SCHEMBL20002698 0.84 HSD11B1 (0.47) EPHX2MEN1ALDH1A1TSHRKMT2A
SCHEMBL20002574 0.84 ALDH1A1 (0.51) EPHX2MEN1ALDH1A1TSHRKMT2A
SCHEMBL20002705 0.84 ALDH1A1 (0.41) MEN1ALDH1A1TSHRKMT2APTPN1
SCHEMBL20002706 0.84 HSD11B1 (0.47) EPHX2MEN1ALDH1A1TSHRKMT2A
SCHEMBL20002746 0.83 CCR5 (0.44) MEN1ALDH1A1TSHRKMT2APTPN1
SCHEMBL20002660 0.82 FASN (0.52) MEN1FASNTSHRKMT2APTPN1
SCHEMBL20003098 0.81 GPR183 (0.38) MEN1ALDH1A1TSHRKMT2APTPN1
SCHEMBL20002995 0.79 GFER (0.50) MEN1ALDH1A1TSHRKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed