SCHEMBL20003098

SCHEMBL20003098

C=Cc1ccc([S+]([O-])C2CCN(C(=O)C3CCCCC3)C2)cc1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GPR183 P32249 1/20 0.38
TSHR P16473 3/20 0.38
ALDH1A1 P00352 2/20 0.38
KMT2A Q03164 4/20 0.37
MEN1 O00255 2/20 0.37
PTPN1 P18031 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.36
KEAP1 Q14145 1/20 0.36
F13A1 P00488 1/20 0.36
TGM2 P21980 1/20 0.36
TGM1 P22735 1/20 0.36
NPSR1 Q6W5P4 2/20 0.36
MAPT P10636 1/20 0.36
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
RIPK1 Q13546 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002641 0.85 TDP1 (0.42) TSHRALDH1A1KMT2AMEN1PTPN1
SCHEMBL20002705 0.84 ALDH1A1 (0.41) TSHRALDH1A1KMT2AMEN1PTPN1
SCHEMBL20002706 0.84 HSD11B1 (0.47) TSHRALDH1A1KMT2AMEN1PTPN1
SCHEMBL20002698 0.84 HSD11B1 (0.47) TSHRALDH1A1KMT2AMEN1PTPN1
SCHEMBL20003089 0.84 GPR183 (0.45) GPR183TSHRALDH1A1KMT2AMEN1
SCHEMBL20002574 0.84 ALDH1A1 (0.51) TSHRALDH1A1KMT2AMEN1SMN1; SMN2
SCHEMBL20002746 0.83 CCR5 (0.44) TSHRALDH1A1KMT2AMEN1PTPN1
SCHEMBL20002660 0.82 FASN (0.52) TSHRKMT2AMEN1PTPN1SMN1; SMN2
SCHEMBL20002932 0.81 KDM1A (0.42) TSHRALDH1A1KMT2AMEN1PTPN1
SCHEMBL20002995 0.79 GFER (0.50) TSHRALDH1A1KMT2AMEN1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed