SCHEMBL20003009

SCHEMBL20003009

O=C(O)C12CCC(C(=O)N3CCC(S(=O)(=O)c4ccc(F)cc4)C3)(CC1)OC2

nearest known ligand 0.54

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
RORC P51449 13/20 0.54
HTR2A P28223 2/20 0.39
HTR2C P28335 1/20 0.39
KCNH2 Q12809 1/20 0.39
EPHX2 P34913 1/20 0.38
GPR6 P46095 1/20 0.38
DRD2 P14416 1/20 0.37
CCR5 P51681 1/20 0.36
NAMPT P43490 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20002497 0.77 RORC (0.44) RORCGPR6CCR5
SCHEMBL20002921 0.76 RORC (0.44) RORCGPR6CCR5
SCHEMBL20002866 0.75 RORC (0.49) RORCHTR2AHTR2CKCNH2EPHX2
SCHEMBL20002828 0.74 RORC (0.54) RORCHTR2AHTR2CKCNH2EPHX2
SCHEMBL20002880 0.73 RORC (0.46) RORCGPR6CCR5
SCHEMBL20002922 0.73 RORC (0.46) RORCEPHX2GPR6CCR5
SCHEMBL20002406 0.73 RORC (0.42) RORCHTR2AHTR2CKCNH2EPHX2
SCHEMBL20002460 0.73 RORC (0.55) RORCHTR2AHTR2CKCNH2EPHX2
SCHEMBL14413535 0.72 EPHX2 (0.47) RORCHTR2AHTR2CKCNH2EPHX2
SCHEMBL20002321 0.72 CCR5 (0.46) RORCEPHX2GPR6CCR5NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed