SCHEMBL20004206

SCHEMBL20004206

COc1cc2c(cc1C)CCC(=O)C2(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 2/20 0.38
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MAPK1 P28482 2/20 0.33
GAA P10253 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC7 Q8WUI4 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC10 Q969S8 1/20 0.33
HDAC11 Q96DB2 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
HDAC9 Q9UKV0 1/20 0.33
HDAC5 Q9UQL6 1/20 0.33
PARP1 P09874 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL897012 0.83 HTR2A (0.45) ALK
SCHEMBL20061137 0.83 S100B (0.38) ALKKMT2AL3MBTL1MAPK1GAA
SCHEMBL897525 0.83 ALK (0.43) ALKMAPK1GAAALDH1A1
SCHEMBL897888 0.81 TAAR1 (0.39) ALKKMT2AMEN1MAPK1ALDH1A1
SCHEMBL20061173 0.79 S100B (0.38) ALKKMT2AL3MBTL1GAAALDH1A1
SCHEMBL29940794 0.79 CHEK1 (0.38) ALKALDH1A1
SCHEMBL7812922 0.79 ALK (0.43) ALKKMT2ASMN1; SMN2ALDH1A1PARP1
SCHEMBL29940534 0.79 ALK (0.38) ALKKMT2AMEN1MAPK1GAA
SCHEMBL27087621 0.79 ALK (0.38) ALKKMT2AMEN1MAPK1GAA
SCHEMBL897548 0.79 CA9 (0.43) ALKKMT2AMEN1MAPK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2975024-B1 TETRACYCLIC COMPOUNDS CHUGAI PHARMACEUTICAL CO LTD (JP) 2018-03-28 EP disclosed