SCHEMBL20004586

SCHEMBL20004586

Cc1ccc(-c2ccc3cc(-c4cc(C)c(C#Cc5ccc(-c6ccc(C)cn6)cc5)cc4F)ccc3c2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 3/20 0.37
PTGS2 P35354 2/20 0.35
CYP11B1 P15538 2/20 0.34
CYP11B2 P19099 2/20 0.34
AAK1 Q2M2I8 1/20 0.33
ABL1 P00519 2/20 0.32
AURKA O14965 1/20 0.32
NTRK1 P04629 1/20 0.32
LCK P06239 1/20 0.32
CSF1R P07333 1/20 0.32
RET P07949 1/20 0.32
MET P08581 1/20 0.32
PDGFRB P09619 1/20 0.32
PIM1 P11309 1/20 0.32
PDGFRA P16234 1/20 0.32
FLT3 P36888 1/20 0.32
MAPK8 P45983 1/20 0.32
CDK8 P49336 1/20 0.32
MAP2K1 Q02750 1/20 0.32
MAP4K2 Q12851 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20004583 0.89 SMN1; SMN2 (0.43) GRM5ABL1AURKANTRK1LCK
SCHEMBL20004879 0.84 FFAR1 (0.34) PTGS2CYP11B1CYP11B2AAK1
SCHEMBL20005287 0.83 ESR1 (0.38) GRM5CYP11B1CYP11B2AAK1
SCHEMBL19999591 0.81 RAB9A (0.42)
SCHEMBL20005267 0.81 RARA (0.39)
SCHEMBL20004894 0.81 RARA (0.39)
SCHEMBL20004878 0.75 HRH3 (0.38)
SCHEMBL20005285 0.74 FFAR1 (0.40)
SCHEMBL20006703 0.73 PDE3B (0.33) GRM5CYP11B1CYP11B2
SCHEMBL20006719 0.73 PDE3B (0.33) GRM5CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3299439-A1 LIQUID CRYSTAL COMPOUND, LIQUID CRYSTAL COMPOSITION AND LIQUID CRYSTAL DISPLAY DEVICE JNC Corporation (JP) 2018-03-28 EP disclosed