SCHEMBL2009494

SCHEMBL2009494

O=C(c1ncc(-c2cccnc2)o1)c1c(Cl)n(Cc2ccc(Cl)cc2Cl)c2ccc(Cl)cc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.37
LMNA P02545 4/20 0.37
ALDH1A1 P00352 3/20 0.37
MAPT P10636 3/20 0.37
ALOX12 P18054 2/20 0.37
KDM4E B2RXH2 2/20 0.37
POLB P06746 1/20 0.37
PKM P14618 1/20 0.37
HPGD P15428 1/20 0.37
TBXAS1 P24557 1/20 0.36
P2RX7 Q99572 1/20 0.35
CYP1A2 P05177 2/20 0.34
CYP2D6 P10635 2/20 0.34
CYP2C9 P11712 2/20 0.34
NPSR1 Q6W5P4 2/20 0.34
CYP3A4 P08684 1/20 0.34
TSHR P16473 1/20 0.34
PMP22 Q01453 1/20 0.34
HIF1A Q16665 1/20 0.34
MEN1 O00255 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2001640 0.95 L3MBTL1 (0.39) FAAHLMNAALDH1A1MAPTALOX12
SCHEMBL2000766 0.94 FAAH (0.36) FAAHLMNAALDH1A1MAPTALOX12
SCHEMBL2005968 0.94 LMNA (0.41) FAAHLMNAALDH1A1MAPTALOX12
SCHEMBL2003366 0.92 TP53 (0.39) FAAHALDH1A1MAPTKDM4EPOLB
SCHEMBL2003027 0.91 POLB (0.37) FAAHLMNAALDH1A1MAPTALOX12
SCHEMBL2002487 0.91 LMNA (0.40) FAAHLMNAALDH1A1MAPTALOX12
SCHEMBL2000331 0.90 PTGES2 (0.41) FAAHLMNAALDH1A1MAPTALOX12
SCHEMBL2006262 0.90 CYP2C9 (0.40) FAAHLMNAALDH1A1MAPTALOX12
SCHEMBL2000666 0.89 PTGES2 (0.35) FAAHLMNAALDH1A1MAPTALOX12
SCHEMBL4389111 0.87 LMNA (0.37) FAAHLMNAALDH1A1MAPTALOX12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed