SCHEMBL20008349

SCHEMBL20008349

C=N/C=C(\C=C/C1CCCCC1)c1cc(NC)ccc1C

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
LDLR P01130 1/20 0.32
NPC1 O15118 2/20 0.32
RAB9A P51151 2/20 0.32
GRIN1 Q05586 1/20 0.31
GRIN2B Q13224 1/20 0.31
TSHR P16473 1/20 0.30
HTT P42858 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
EPHX2 P34913 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20008807 0.87 LDLR (0.31) LDLRNPC1RAB9AGRIN1GRIN2B
SCHEMBL20008589 0.83 GRIN1 (0.34) GRIN1GRIN2BTSHR
SCHEMBL20008490 0.81 PLAU (0.32)
SCHEMBL22561935 0.71
SCHEMBL22561986 0.69 LDLR (0.33) LDLRNPC1RAB9A
SCHEMBL20008372 0.63 OPRK1 (0.31)
SCHEMBL20009063 0.63 NPC1 (0.39) NPC1RAB9AHTTSMN1; SMN2
SCHEMBL20008487 0.62 NPC1 (0.36) NPC1RAB9AHTTSMN1; SMN2
SCHEMBL20009403 0.62
SCHEMBL20008186 0.62

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3299367-A1 BIARYL AMIDE COMPOUNDS AS KINASE INHIBITORS Novartis AG (CH) 2018-03-28 EP disclosed