SCHEMBL20008589

SCHEMBL20008589

C=N/C=C(\C=C/C1CCCCC1)c1cc(N)ccc1C

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 1/20 0.34
GRIN2B Q13224 1/20 0.34
TSHR P16473 1/20 0.31
CASP1 P29466 1/20 0.31
GFER P55789 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20008349 0.83 LDLR (0.32) GRIN1GRIN2BTSHR
SCHEMBL20008807 0.70 LDLR (0.31) GRIN1GRIN2B
SCHEMBL25992719 0.65 CASP1 (0.40) TSHRCASP1ALDH1A1
SCHEMBL14964429 0.64 ALDH1A1 (0.52) TSHRCASP1ALDH1A1
SCHEMBL22562067 0.62 CYP2D6 (0.40)
SCHEMBL20076793 0.59 ALDH1A1 (0.56) TSHRCASP1ALDH1A1
SCHEMBL21020629 0.59 ALDH1A1 (0.50) TSHRCASP1ALDH1A1
SCHEMBL20008147 0.59 CASP1 (0.35) TSHRCASP1ALDH1A1
SCHEMBL26084626 0.58 CASP1 (0.37) TSHRCASP1ALDH1A1
SCHEMBL23525688 0.57 CYP19A1 (0.44) TSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3299367-A1 BIARYL AMIDE COMPOUNDS AS KINASE INHIBITORS Novartis AG (CH) 2018-03-28 EP disclosed