SCHEMBL22561986

SCHEMBL22561986

C=N/C=C(\C=C(\C#N)C1CCCCC1)c1cc(N/C(C)=C\C)ccc1C

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
LDLR P01130 1/20 0.33
NPC1 O15118 2/20 0.31
RAB9A P51151 2/20 0.31
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
HPGD P15428 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22562067 0.78 CYP2D6 (0.40)
SCHEMBL22561935 0.70
SCHEMBL22561885 0.65 GABRA1 (0.38)
SCHEMBL20008807 0.59 LDLR (0.31) LDLRNPC1RAB9A
SCHEMBL22561897 0.56
SCHEMBL24060059 0.55 RAB9A (0.72) NPC1RAB9AKDM4EALDH1A1HPGD
SCHEMBL14435612 0.53 MGLL (0.37) LDLRNPC1RAB9AALDH1A1
SCHEMBL24746313 0.53 NPC1 (0.62) NPC1RAB9AKDM4EALDH1A1
SCHEMBL26145831 0.53 HPGD (0.51) NPC1RAB9AKDM4EALDH1A1HPGD
SCHEMBL18664789 0.52 ALDH1A1 (0.60) NPC1RAB9AKDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3191467-B1 COMPOUNDS AND COMPOSITIONS AS KINASE INHIBITORS NOVARTIS AG (CH) 2020-10-21 EP disclosed