SCHEMBL20009063

SCHEMBL20009063

CN/C=C(\C=C(/C)N1CCCCC1)c1cc(NC)ccc1C

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.39
RAB9A P51151 4/20 0.39
MAPT P10636 1/20 0.36
HTT P42858 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
USP2 O75604 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
ALOX12 P18054 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
KMT2A Q03164 2/20 0.33
TP53 P04637 1/20 0.33
MEN1 O00255 1/20 0.33
FKBP1A P62942 1/20 0.32
TDP1 Q9NUW8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20008363 0.99 MAPT (0.37) NPC1RAB9AMAPTHTTL3MBTL1
SCHEMBL20008487 0.89 NPC1 (0.36) NPC1RAB9AMAPTHTTL3MBTL1
SCHEMBL20008164 0.85 MAPT (0.32) NPC1RAB9AMAPTHTTL3MBTL1
SCHEMBL20009507 0.81 MAPT (0.33) MAPTUSP2ALDH1A1LMNAALOX12
SCHEMBL20008254 0.79 NPC1 (0.34) NPC1RAB9AHTTL3MBTL1ALDH1A1
SCHEMBL20009408 0.77 BRAF (0.45) NPC1RAB9AMAPTHTTUSP2
SCHEMBL20008383 0.76 MAPT (0.38) NPC1RAB9AMAPTHTTL3MBTL1
SCHEMBL20008308 0.73 NPC1 (0.36) NPC1RAB9AHTTL3MBTL1SMN1; SMN2
SCHEMBL20008233 0.72 RAB9A (0.39) NPC1RAB9AMAPTHTTL3MBTL1
SCHEMBL20008169 0.71 PABPC1 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3299367-A1 BIARYL AMIDE COMPOUNDS AS KINASE INHIBITORS Novartis AG (CH) 2018-03-28 EP disclosed