SCHEMBL20009541

SCHEMBL20009541

C=CCCC/C(N)=C(/C=C(\N)c1cc(C)ccc1C)N1CCCC1

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.32
DRD2 P14416 2/20 0.31
DRD4 P21917 2/20 0.31
DRD3 P35462 2/20 0.31
RAB9A P51151 2/20 0.31
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
TSHR P16473 1/20 0.30
CYP2D6 P10635 1/20 0.30
NPC1 O15118 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19529299 0.69 SMN1; SMN2 (0.41) RAB9ASMN1; SMN2CYP2D6NPC1
SCHEMBL20008464 0.66 NPC1 (0.30) RAB9AKMT2ANPC1
SCHEMBL20008233 0.65 RAB9A (0.39) TP53RAB9AKMT2ASMN1; SMN2NPC1
SCHEMBL25464953 0.64 CYP2D6 (0.40) TP53MEN1KMT2ASMN1; SMN2TSHR
SCHEMBL20008581 0.63 TP53 (0.39) TP53DRD2DRD4DRD3RAB9A
SCHEMBL20008429 0.61 TP53 (0.40) TP53RAB9AMEN1KMT2ASMN1; SMN2
SCHEMBL12846473 0.61 HPGD (0.58) RAB9AMEN1KMT2ATSHRNPC1
SCHEMBL20008272 0.61 TP53 (0.40) TP53RAB9AMEN1KMT2ASMN1; SMN2
SCHEMBL15306495 0.60 HPGD (0.57) TP53RAB9AMEN1KMT2ASMN1; SMN2
SCHEMBL20008223 0.58 TP53 (0.39) TP53RAB9AMEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3299367-A1 BIARYL AMIDE COMPOUNDS AS KINASE INHIBITORS Novartis AG (CH) 2018-03-28 EP disclosed