SCHEMBL20011251

SCHEMBL20011251

Cc1cc(CCCCn2c(=O)c3c(n(C)c2=O)NCN3C)no1

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 2/20 0.36
GRIN1 Q05586 8/20 0.35
GRIN2B Q13224 8/20 0.35
PARG Q86W56 2/20 0.34
GABRA5 P31644 2/20 0.33
MAPT P10636 1/20 0.33
RECQL P46063 1/20 0.33
GABRA1 P14867 1/20 0.32
NMT1 P30419 2/20 0.31
TNF P01375 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20011175 0.80 PARG (0.31) PARGTNF
SCHEMBL20011542 0.73 TNF (0.35) TNF
SCHEMBL4557788 0.72 TNF (0.46) MAPTTNF
SCHEMBL18255777 0.72 ADORA2B (0.58) TRPA1TNF
SCHEMBL17619749 0.72 TRPA1 (0.57) TRPA1GRIN1GRIN2BPARGGABRA5
SCHEMBL20011328 0.72 PARG (0.33) PARG
SCHEMBL17619786 0.70 TRPA1 (0.58) TRPA1GRIN1GRIN2BPARG
SCHEMBL20011548 0.69 PARG (0.33) PARG
SCHEMBL18256158 0.69 TRPA1 (0.52) TRPA1MAPTTNF
SCHEMBL20011545 0.68 PARG (0.41) GRIN1GRIN2BPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3299371-A1 HYDROXYL PURINE COMPOUNDS AND USE THEREOF GUANGDONG ZHONGSHENG PHARMACEUTICAL CO., LTD (CN) 2018-03-28 EP disclosed