SCHEMBL2001648

SCHEMBL2001648

O=C(c1noc(-c2ccncc2)n1)c1c(C(F)(F)F)n(Cc2ccc(Cl)cc2Cl)c2ccc(Cl)cc12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RET P07949 1/20 0.37
CYP3A4 P08684 2/20 0.36
CYP2C9 P11712 2/20 0.36
ROCK2 O75116 1/20 0.35
ROCK1 Q13464 1/20 0.35
SRPK1 Q96SB4 1/20 0.34
LMNA P02545 4/20 0.34
TSHR P16473 3/20 0.34
MAPK1 P28482 2/20 0.34
TAAR1 Q96RJ0 1/20 0.34
GSK3A P49840 1/20 0.34
GSK3B P49841 1/20 0.34
KMT2A Q03164 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
ALOX12 P18054 1/20 0.34
CASP1 P29466 1/20 0.34
RAB9A P51151 2/20 0.33
DUSP3 P51452 1/20 0.33
PTPN11 Q06124 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2003892 0.95 L3MBTL1 (0.36) RETCYP3A4CYP2C9ROCK2ROCK1
SCHEMBL2008461 0.94 RET (0.36) RETCYP3A4CYP2C9ROCK2ROCK1
SCHEMBL2012645 0.93 LMNA (0.40) RETCYP3A4CYP2C9ROCK2ROCK1
SCHEMBL2001214 0.92 PLA2G2A (0.38) RETCYP3A4CYP2C9LMNATSHR
SCHEMBL2002572 0.91 HSD17B10 (0.36) RETCYP3A4CYP2C9SRPK1TSHR
SCHEMBL2003150 0.91 S1PR1 (0.35) RETCYP3A4CYP2C9SRPK1LMNA
SCHEMBL2004314 0.90 RET (0.39) RETLMNATSHRMAPK1ALDH1A1
SCHEMBL1999738 0.89 CYP2C9 (0.39) CYP3A4CYP2C9ROCK2ROCK1LMNA
SCHEMBL2005893 0.89 SCD (0.34) CYP3A4CYP2C9ROCK2ROCK1LMNA
SCHEMBL2004941 0.86 GRM5 (0.38) CYP3A4CYP2C9LMNATSHRKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed