SCHEMBL2008461

SCHEMBL2008461

Cc1ccc2c(c1)c(C(=O)c1noc(-c3ccncc3)n1)c(C(F)(F)F)n2Cc1ccc(Cl)cc1Cl

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RET P07949 1/20 0.36
NPC1 O15118 2/20 0.34
RAB9A P51151 1/20 0.34
CYP3A4 P08684 2/20 0.33
CYP2C9 P11712 2/20 0.33
SRPK1 Q96SB4 1/20 0.33
ROCK2 O75116 1/20 0.33
ROCK1 Q13464 1/20 0.33
HSD17B10 Q99714 1/20 0.33
LMNA P02545 3/20 0.32
MAPK1 P28482 2/20 0.32
KMT2A Q03164 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
TAAR1 Q96RJ0 1/20 0.32
TSHR P16473 1/20 0.32
GSK3A P49840 1/20 0.32
GSK3B P49841 1/20 0.32
FAAH O00519 1/20 0.32
TP53 P04637 2/20 0.32
KDM4E B2RXH2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2001648 0.94 RET (0.37) RETNPC1RAB9ACYP3A4CYP2C9
SCHEMBL2003892 0.91 L3MBTL1 (0.36) RETNPC1RAB9ACYP3A4CYP2C9
SCHEMBL2006095 0.91 FAAH (0.39) CYP3A4CYP2C9SRPK1HSD17B10KMT2A
SCHEMBL2002558 0.91 RET (0.39) RETNPC1RAB9ALMNAMAPK1
SCHEMBL2001214 0.90 PLA2G2A (0.38) RETNPC1RAB9ACYP3A4CYP2C9
SCHEMBL2012645 0.90 LMNA (0.40) RETCYP3A4CYP2C9SRPK1ROCK2
SCHEMBL2004301 0.90 RAB9A (0.36) NPC1RAB9ACYP3A4CYP2C9ROCK2
SCHEMBL2009499 0.89 FAAH (0.33) NPC1CYP3A4CYP2C9LMNAMAPK1
SCHEMBL2003150 0.89 S1PR1 (0.35) RETCYP3A4CYP2C9SRPK1HSD17B10
SCHEMBL2006492 0.87 GRM5 (0.35) NPC1CYP3A4CYP2C9LMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed