SCHEMBL20021168

SCHEMBL20021168

NCc1ccc2c3c(cccc13)CCO2

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCI P41743 1/20 0.37
MAPT P10636 2/20 0.35
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
GAA P10253 1/20 0.35
HPGD P15428 1/20 0.35
KMT2A Q03164 1/20 0.35
DYRK1A Q13627 3/20 0.35
PARP1 P09874 1/20 0.34
CD274 Q9NZQ7 1/20 0.34
AURKA O14965 1/20 0.34
RPS6KB1 P23443 1/20 0.34
RAB9A P51151 2/20 0.33
NPC1 O15118 1/20 0.33
POLB P06746 1/20 0.33
DYRK2 Q92630 1/20 0.33
DYRK1B Q9Y463 1/20 0.33
KEAP1 Q14145 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20021160 0.84 PRKCI (0.34) PRKCIMAPTKDM4EMEN1ALDH1A1
SCHEMBL20020909 0.84 KDM4E (0.38) PRKCIMAPTKDM4EALDH1A1HPGD
SCHEMBL5165673 0.78 KDM4E (0.57) MAPTKDM4EMEN1ALDH1A1LMNA
SCHEMBL3298420 0.76 TYMS (0.45) PRKCIMAPTKDM4EMEN1ALDH1A1
SCHEMBL15182506 0.72 FABP4 (0.35) PRKCIMAPTKDM4EMEN1ALDH1A1
SCHEMBL20021100 0.72 HPGD (0.44) PRKCIMAPTKDM4EMEN1ALDH1A1
SCHEMBL13736784 0.72 KEAP1 (0.38) PRKCIKDM4EMEN1ALDH1A1HPGD
SCHEMBL1150915 0.69 PARP1 (0.51) PARP1PNMT
SCHEMBL21662885 0.69 CYP3A4 (0.41) PRKCIMAPTKDM4EALDH1A1LMNA
SCHEMBL28860523 0.68 PNMT (0.44) MEN1KMT2APARP1CD274PNMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2588455-B1 2-QUINOLINYL-ACETIC ACID DERIVATIVES AS HIV ANTIVIRAL COMPOUNDS GILEAD SCIENCES INC (US) 2018-04-04 EP disclosed