SCHEMBL20027641

SCHEMBL20027641

CNNc1cccc(CO)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.46
PDK2 Q15119 1/20 0.46
PDK3 Q15120 1/20 0.46
PDK4 Q16654 1/20 0.46
TOP2A P11388 1/20 0.45
TOP2B Q02880 1/20 0.45
IKBKB O14920 1/20 0.44
ALDH1A1 P00352 3/20 0.43
ENPP2 Q13822 1/20 0.42
ABCG2 Q9UNQ0 1/20 0.42
SYK P43405 1/20 0.41
FLT1 P17948 1/20 0.40
FLT4 P35916 1/20 0.40
KDR P35968 1/20 0.40
PRSS1 P07477 1/20 0.40
PRSS2 P07478 1/20 0.40
PRSS3 P35030 1/20 0.40
TSHR P16473 1/20 0.39
PRKCI P41743 1/20 0.39
KDM1A O60341 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3150743 0.83 PDK1 (0.49) PDK1PDK2PDK3PDK4TOP2A
SCHEMBL16590399 0.82 RAPGEF4 (0.51) ALDH1A1MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL20027769 0.80 HTR6 (0.47) ALDH1A1ENPP2SMN1; SMN2
SCHEMBL27815971 0.80 PDK1 (0.46) PDK1PDK2PDK3PDK4TOP2A
SCHEMBL7258875 0.77 ALDH1A1 (0.47) ALDH1A1KDRTSHRKDM1ARCOR1
SCHEMBL10708264 0.77 TOP2A (0.49) PDK1PDK2PDK3PDK4TOP2A
SCHEMBL3103338 0.76 PDK1 (0.46) PDK1PDK2PDK3PDK4TOP2A
SCHEMBL23197732 0.76 NOS3 (0.35) PDK1PDK2PDK3PDK4MAPT
SCHEMBL4354231 0.75 TOP2A (0.47) PDK1PDK2PDK3PDK4TOP2A
SCHEMBL3103283 0.74 TDP1 (0.48) PDK1PDK2PDK3PDK4TOP2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018064119-A1 CALPAIN MODULATORS AND THERAPEUTIC USES THEREOF BLADE THERAPEUTICS, INC. (US) 2018-04-05 WO disclosed