SCHEMBL2002947

SCHEMBL2002947

Cc1ccc2c(c1)c(C(=O)c1ncc(-c3ccncc3)o1)c(C(F)(F)F)n2Cc1ccc(Cl)cc1Cl

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
FAAH O00519 2/20 0.33
PTGS1 P23219 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
NPC1 O15118 1/20 0.33
LMNA P02545 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
TAAR1 Q96RJ0 1/20 0.32
RIPK3 Q9Y572 1/20 0.32
TP53 P04637 1/20 0.32
MAPK1 P28482 1/20 0.32
CASP1 P29466 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
ALOX12 P18054 1/20 0.31
F10 P00742 1/20 0.31
SLC26A4 O43511 1/20 0.31
POLB P06746 1/20 0.31
EPHX2 P34913 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2006841 0.94 CYP3A4 (0.37) CYP3A4CYP2C9FAAHNPC1LMNA
SCHEMBL2005400 0.93 PPARG (0.36) CYP3A4CYP2C9FAAHPTGS1PTGDR2
SCHEMBL2004824 0.92 PTGES2 (0.36) CYP2C9FAAHPTGS1PTGDR2NPC1
SCHEMBL2005377 0.92 L3MBTL1 (0.36) CYP3A4CYP2C9FAAHLMNATAAR1
SCHEMBL2005131 0.91 FAAH (0.41) CYP3A4CYP2C9FAAHPTGDR2MAPT
SCHEMBL2004961 0.90 FAAH (0.33) FAAHPTGS1PTGDR2NPC1LMNA
SCHEMBL2008690 0.90 PLA2G2A (0.38) CYP3A4CYP2C9PTGDR2LMNATP53
SCHEMBL2003600 0.90 LMNA (0.40) CYP3A4CYP2C9LMNASMN1; SMN2TAAR1
SCHEMBL2006660 0.90 CYP2C9 (0.37) CYP3A4CYP2C9FAAHPTGS1PTGDR2
SCHEMBL1999823 0.90 F2RL3 (0.36) CYP3A4CYP2C9LMNASMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed