SCHEMBL2008690

SCHEMBL2008690

COc1ccc2c(c1)c(C(=O)c1ncc(-c3ccncc3)o1)c(C(F)(F)F)n2Cc1ccc(Cl)cc1Cl

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLA2G2A P14555 4/20 0.38
PTGS2 P35354 1/20 0.36
F2RL3 Q96RI0 4/20 0.36
CYP3A4 P08684 4/20 0.35
CYP2C9 P11712 4/20 0.35
CYP1A2 P05177 3/20 0.35
CYP2D6 P10635 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35
TP53 P04637 2/20 0.35
MAPT P10636 2/20 0.35
SLC26A4 O43511 1/20 0.34
POLB P06746 1/20 0.34
GSK3B P49841 1/20 0.34
SRPK1 Q96SB4 1/20 0.34
F10 P00742 1/20 0.34
MEN1 O00255 1/20 0.33
RGS12 O14924 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
PKM P14618 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1999823 0.93 F2RL3 (0.36) F2RL3CYP3A4CYP2C9CYP1A2CYP2D6
SCHEMBL2004514 0.93 F2RL3 (0.39) PLA2G2APTGS2F2RL3CYP3A4CYP2C9
SCHEMBL2006841 0.92 CYP3A4 (0.37) CYP3A4CYP2C9CYP1A2CYP2D6MAPT
SCHEMBL2001047 0.92 PLA2G2A (0.37) PLA2G2APTGS2F2RL3CYP3A4CYP2C9
SCHEMBL1998915 0.91 LMNA (0.42) PLA2G2APTGS2CYP3A4CYP2C9CYP1A2
SCHEMBL2010346 0.91 PLA2G2A (0.37) PLA2G2APTGS2F2RL3CYP3A4CYP2C9
SCHEMBL2002947 0.90 CYP3A4 (0.35) CYP3A4CYP2C9PTGDR2TP53MAPT
SCHEMBL2004240 0.90 PLA2G2A (0.39) PLA2G2ACYP3A4CYP2C9CYP1A2PTGDR2
SCHEMBL2005377 0.89 L3MBTL1 (0.36) CYP3A4CYP2C9MAPTGSK3BF10
SCHEMBL2000385 0.88 FAAH (0.38) PLA2G2AF2RL3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed