SCHEMBL1996791

SCHEMBL1996791

Cc1ccc2c(c1)c(C(=O)c1cnc(-c3cccnc3)o1)c(Cl)n2Cc1ccc(Cl)cc1Cl

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES2 Q9H7Z7 1/20 0.38
TBXAS1 P24557 1/20 0.37
MAPT P10636 4/20 0.37
ALDH1A1 P00352 3/20 0.37
ALOX12 P18054 3/20 0.37
NPSR1 Q6W5P4 3/20 0.37
KDM4E B2RXH2 2/20 0.37
HPGD P15428 2/20 0.37
ALOX15 P16050 1/20 0.37
HSD17B10 Q99714 1/20 0.37
FAAH O00519 1/20 0.37
LMNA P02545 3/20 0.36
POLB P06746 1/20 0.36
PKM P14618 1/20 0.36
P2RX7 Q99572 1/20 0.36
ALOX5AP P20292 1/20 0.35
HDAC1 Q13547 2/20 0.34
HDAC6 Q9UBN7 2/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2003941 0.94 P2RX7 (0.38) PTGES2TBXAS1MAPTALDH1A1ALOX12
SCHEMBL2008233 0.92 LMNA (0.39) PTGES2MAPTALDH1A1ALOX12NPSR1
SCHEMBL2002956 0.92 PTGES2 (0.44) PTGES2TBXAS1MAPTALDH1A1ALOX12
SCHEMBL2002287 0.91 L3MBTL1 (0.39) PTGES2TBXAS1MAPTALDH1A1ALOX12
SCHEMBL2012281 0.91 FAAH (0.38) MAPTALDH1A1ALOX12NPSR1KDM4E
SCHEMBL2008737 0.91 LMNA (0.42) TBXAS1MAPTALDH1A1ALOX12NPSR1
SCHEMBL2006372 0.90 PTGES2 (0.39) PTGES2TBXAS1MAPTALDH1A1ALOX12
SCHEMBL2003889 0.90 ALDH1A1 (0.38) MAPTALDH1A1KDM4EHPGDLMNA
SCHEMBL2006172 0.89 ALOX5AP (0.39) PTGES2MAPTKDM4ELMNAPOLB
SCHEMBL2006623 0.87 POLB (0.38) PTGES2TBXAS1MAPTALDH1A1ALOX12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed