SCHEMBL2003586

SCHEMBL2003586

Cc1ccc2c(c1)c(C(=O)c1noc(-c3ccccc3)n1)c(Cl)n2Cc1ccc(Cl)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
HTT P42858 1/20 0.42
PTGES2 Q9H7Z7 4/20 0.42
PTGES O14684 2/20 0.42
FAAH O00519 1/20 0.41
DRD2 P14416 1/20 0.40
CNR2 P34972 2/20 0.40
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 1/20 0.39
GAA P10253 1/20 0.39
HSD17B10 Q99714 1/20 0.39
PPARG P37231 1/20 0.39
AKR1B1 P15121 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
DHODH Q02127 1/20 0.38
ALOX5 P09917 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1999518 0.93 MAPT (0.43) KMT2AMEN1HTTPTGES2PTGES
SCHEMBL2002667 0.92 MEN1 (0.42) KMT2AMEN1HTTFAAHDRD2
SCHEMBL2004165 0.90 LMNA (0.38) KMT2ALMNAMAPTALDH1A1KDM4E
SCHEMBL2001735 0.90 MAPT (0.42) KMT2AMEN1PTGES2PTGESDRD2
SCHEMBL2006486 0.89 PTGES2 (0.41) KMT2AMEN1HTTPTGES2PTGES
SCHEMBL2005851 0.89 ALDH1A1 (0.43) KMT2AMEN1HTTPTGES2DRD2
SCHEMBL2001661 0.89 PLA2G2A (0.48) KMT2AMEN1LMNAMAPTALDH1A1
SCHEMBL2006918 0.88 FAAH (0.44) KMT2AMEN1HTTFAAHMAPT
SCHEMBL2003154 0.87 ALOX5AP (0.42) KMT2AMAPTSMN1; SMN2ALOX5
SCHEMBL2003864 0.84 MAPT (0.38) KMT2AMEN1FAAHDRD2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed