SCHEMBL2003162

SCHEMBL2003162

COc1ccc2c(c1)c(C(=O)c1nc(-c3ccncn3)no1)c(C(F)(F)F)n2Cc1ccc(Cl)cc1Cl

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLA2G2A P14555 3/20 0.37
PTGS2 P35354 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.34
TP53 P04637 2/20 0.33
MAPT P10636 5/20 0.33
PPARG P37231 1/20 0.33
ALOX5AP P20292 1/20 0.32
LMNA P02545 3/20 0.32
CYP2C9 P11712 3/20 0.32
ALDH1A1 P00352 2/20 0.32
MAPK1 P28482 2/20 0.32
CYP1A2 P05177 2/20 0.32
CYP3A4 P08684 2/20 0.32
MEN1 O00255 1/20 0.32
RGS12 O14924 1/20 0.32
PKM P14618 1/20 0.32
TSHR P16473 1/20 0.32
NFKB1 P19838 1/20 0.32
CYP2C19 P33261 1/20 0.32
GNAI1 P63096 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2002732 0.94 LMNA (0.33) PLA2G2APTGS2MAPTALOX5APLMNA
SCHEMBL2005062 0.94 EPHX2 (0.33) TP53MAPTLMNACYP2C9ALDH1A1
SCHEMBL2005516 0.91 FAAH (0.33) PTGDR2TP53LMNACYP2C9MAPK1
SCHEMBL2004491 0.91 LMNA (0.41) PLA2G2APTGS2MAPTALOX5APLMNA
SCHEMBL4564522 0.91 NPC1 (0.38) PLA2G2APTGS2TP53MAPTALOX5AP
SCHEMBL2007750 0.91 L3MBTL1 (0.34) TP53MAPTLMNAALDH1A1TSHR
SCHEMBL2003124 0.91 PLA2G2A (0.37) PLA2G2APTGDR2TP53MAPTALOX5AP
SCHEMBL2003311 0.90 PLA2G2A (0.42) PLA2G2APTGS2PTGDR2MAPTPPARG
SCHEMBL2007930 0.90 PLA2G2A (0.38) PLA2G2APTGS2TP53MAPTLMNA
SCHEMBL2007450 0.89 LMNA (0.38) TP53MAPTLMNACYP2C9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed