SCHEMBL20042671

SCHEMBL20042671

Cc1nc2c(c(N3CCC3)n1)CN(C(=O)c1ccc(C)c(C)c1)C2

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.45
ALDH1A1 P00352 4/20 0.44
TSHR P16473 3/20 0.44
HPGD P15428 3/20 0.44
TP53 P04637 1/20 0.44
HTT P42858 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
CNR1 P21554 1/20 0.40
CNR2 P34972 1/20 0.40
GPR55 Q9Y2T6 1/20 0.40
GBA1 P04062 3/20 0.39
PLA2G7 Q13093 1/20 0.38
GAA P10253 1/20 0.37
KMT2A Q03164 1/20 0.37
PRLHR P49683 2/20 0.37
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042752 0.91 HPGD (0.47) P2RX7ALDH1A1TSHRHPGDTP53
SCHEMBL20042823 0.90 P2RX7 (0.45) P2RX7ALDH1A1TSHRHPGDHTT
SCHEMBL20042836 0.90 P2RX7 (0.43) P2RX7ALDH1A1TSHRHPGDTP53
SCHEMBL20042887 0.90 GPR6 (0.42) P2RX7ALDH1A1TSHRHPGDTP53
SCHEMBL20042903 0.88 MEN1 (0.42) P2RX7ALDH1A1TSHRHPGDNPSR1
SCHEMBL20042817 0.87 PKM (0.44) P2RX7ALDH1A1HPGDGBA1KMT2A
SCHEMBL20042666 0.87 KMT2A (0.46) P2RX7CNR1CNR2GPR55GBA1
SCHEMBL20042886 0.87 HPGD (0.49) P2RX7TSHRHPGDKMT2A
SCHEMBL20042872 0.85 P2RX7 (0.44) P2RX7SMN1; SMN2CNR1CNR2GPR55
SCHEMBL20042668 0.85 HPGD (0.51) P2RX7ALDH1A1HPGDHTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed