SCHEMBL20042685

SCHEMBL20042685

Cc1nc2c(c(N3CCC3)n1)CN(C(=O)c1ccc(F)cc1)C2

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.42
P2RX7 Q99572 2/20 0.42
ABL1 P00519 1/20 0.42
BCR P11274 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
TACR3 P29371 2/20 0.41
CYP2C19 P33261 2/20 0.41
CYP2C9 P11712 1/20 0.41
KCNH2 Q12809 1/20 0.41
GBA1 P04062 3/20 0.40
EPHX2 P34913 1/20 0.39
HSD11B1 P28845 1/20 0.39
CYP1A2 P05177 1/20 0.39
GRM5 P41594 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
SLC6A7 Q99884 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042817 0.91 PKM (0.44) P2RX7GBA1SLC6A7
SCHEMBL20042751 0.88 HSD17B10 (0.49) HTTP2RX7TACR3KCNH2GBA1
SCHEMBL20042829 0.88 P2RX7 (0.41) HTTP2RX7TACR3KCNH2GBA1
SCHEMBL20042839 0.88 P2RX7 (0.45) HTTP2RX7L3MBTL1GBA1SMN1; SMN2
SCHEMBL20042704 0.88 P2RX7 (0.50) HTTP2RX7ABL1BCRCYP2C19
SCHEMBL20042666 0.88 KMT2A (0.46) P2RX7TACR3KCNH2GBA1HSD11B1
SCHEMBL20042823 0.87 P2RX7 (0.45) HTTP2RX7TACR3GBA1HSD11B1
SCHEMBL20042836 0.87 P2RX7 (0.43) HTTP2RX7TACR3GBA1SMN1; SMN2
SCHEMBL20042684 0.87 SMN1; SMN2 (0.52) HTTP2RX7ABL1BCRCYP2C19
SCHEMBL20042728 0.85 MEN1 (0.42) L3MBTL1GBA1EPHX2SLC6A7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed