SCHEMBL20042680

SCHEMBL20042680

COc1ccc(C(=O)N2Cc3nc(C)nc(N4CCC4)c3C2)cc1Cl

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR6 P46095 1/20 0.44
TP53 P04637 2/20 0.43
HPGD P15428 4/20 0.42
LRRK2 Q5S007 4/20 0.42
MAPT P10636 5/20 0.41
LMNA P02545 3/20 0.41
ALDH1A1 P00352 4/20 0.40
TAS1R3 Q7RTX0 1/20 0.40
TAS1R1 Q7RTX1 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
KDM4E B2RXH2 2/20 0.39
MAPK1 P28482 2/20 0.39
MALT1 Q9UDY8 1/20 0.39
P2RX7 Q99572 1/20 0.39
GAA P10253 1/20 0.39
ATM Q13315 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TSHR P16473 1/20 0.39
CASP1 P29466 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042752 0.89 HPGD (0.47) TP53HPGDMAPTLMNAALDH1A1
SCHEMBL20042886 0.89 HPGD (0.49) GPR6HPGDKMT2AP2RX7TSHR
SCHEMBL20042911 0.89 P2RX7 (0.39) GPR6TP53HPGDLRRK2MAPT
SCHEMBL20042765 0.89 P2RX7 (0.42) GPR6HPGDLRRK2MALT1P2RX7
SCHEMBL20042700 0.87 TSHR (0.40) TP53HPGDLRRK2MAPTLMNA
SCHEMBL20042667 0.86 TACR3 (0.46) P2RX7
SCHEMBL20042887 0.86 GPR6 (0.42) GPR6TP53HPGDMAPTALDH1A1
SCHEMBL20042733 0.84 MEN1 (0.41) HPGDALDH1A1MEN1KMT2AKDM4E
SCHEMBL20042792 0.84 TACR3 (0.46) GPR6TP53HPGDMAPTMEN1
SCHEMBL20042880 0.83 P2RX7 (0.40) HPGDLRRK2MAPTLMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed