SCHEMBL20042720

SCHEMBL20042720

Cc1nc2c(c(N3CCC3)n1)CN(C(=O)c1cnc(C)c(Cl)c1)C2

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 9/20 0.41
HSP90AA1 P07900 2/20 0.39
P2RX7 Q99572 3/20 0.36
CXCR3 P49682 1/20 0.35
HSP90AB1 P08238 1/20 0.35
P2RY12 Q9H244 5/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042756 0.89 P2RX7 (0.38) HSP90AA1P2RX7
SCHEMBL20042769 0.88 P2RX7 (0.38) HSP90AA1P2RX7
SCHEMBL20042752 0.85 HPGD (0.47) P2RX7
SCHEMBL20042886 0.85 HPGD (0.49) P2RX7
SCHEMBL20042674 0.84 P2RX7 (0.37) HSP90AA1P2RX7
SCHEMBL20042689 0.84 P2RX7 (0.39) GRM5HSP90AA1P2RX7
SCHEMBL20042700 0.83 TSHR (0.40) HSP90AA1P2RX7
SCHEMBL20042667 0.82 TACR3 (0.46) P2RX7
SCHEMBL20042887 0.82 GPR6 (0.42) P2RX7
SCHEMBL20042755 0.82 GRM5 (0.43) GRM5P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed