SCHEMBL20042689

SCHEMBL20042689

Cc1nc2c(c(N3CCC3)n1)CN(C(=O)c1cc(Cl)cc(Cl)c1)C2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 4/20 0.39
TP53 P04637 1/20 0.37
THRB P10828 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
GBA1 P04062 3/20 0.36
CNR2 P34972 1/20 0.36
HSD17B10 Q99714 1/20 0.36
GRM5 P41594 1/20 0.36
PROKR1 Q8TCW9 1/20 0.35
HSP90AA1 P07900 1/20 0.35
FABP3 P05413 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
FABP4 P15090 1/20 0.35
FABP5 Q01469 1/20 0.35
ENPP2 Q13822 1/20 0.35
MAPT P10636 1/20 0.34
USP2 O75604 1/20 0.34
CASP1 P29466 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042854 0.94 GRM5 (0.42) P2RX7TP53THRBTDP1GBA1
SCHEMBL20042863 0.92 GRM5 (0.42) P2RX7TP53THRBTDP1GBA1
SCHEMBL20042702 0.90 P2RX7 (0.49) P2RX7CNR2HSD17B10CYP3A4CYP2D6
SCHEMBL20042656 0.90 KDM4E (0.37) P2RX7TP53THRBTDP1HSD17B10
SCHEMBL20042771 0.89 P2RX7 (0.47) P2RX7GRM5HSP90AA1CYP3A4MAPT
SCHEMBL20042674 0.89 P2RX7 (0.37) P2RX7TP53THRBTDP1GBA1
SCHEMBL20042751 0.88 HSD17B10 (0.49) P2RX7GBA1HSD17B10USP2CASP1
SCHEMBL20042743 0.88 P2RX7 (0.40) P2RX7GBA1CNR2HSD17B10PROKR1
SCHEMBL20042861 0.87 P2RX7 (0.39) P2RX7HSD17B10GRM5MAPTCASP1
SCHEMBL20042829 0.86 P2RX7 (0.41) P2RX7GBA1CNR2HSD17B10GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed