SCHEMBL20042756

SCHEMBL20042756

Cc1nc2c(c(N3CCC3)n1)CN(C(=O)c1cnc(C)c(C)c1)C2

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.38
GPR55 Q9Y2T6 4/20 0.35
CNR1 P21554 4/20 0.35
CNR2 P34972 1/20 0.35
GBA1 P04062 5/20 0.34
HSP90AA1 P07900 3/20 0.33
KMT2A Q03164 3/20 0.33
TSHR P16473 2/20 0.33
MEN1 O00255 2/20 0.33
LMNA P02545 1/20 0.33
NR4A1 P22736 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 2/20 0.33
HTT P42858 1/20 0.33
HSP90B1 P14625 1/20 0.32
MAPK1 P28482 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042720 0.89 GRM5 (0.41) P2RX7HSP90AA1
SCHEMBL20042769 0.89 P2RX7 (0.38) P2RX7GPR55CNR1CNR2GBA1
SCHEMBL20042671 0.84 P2RX7 (0.45) P2RX7GPR55CNR1CNR2GBA1
SCHEMBL20042755 0.83 GRM5 (0.43) P2RX7GBA1KMT2ATSHRMEN1
SCHEMBL20042873 0.83 P2RX7 (0.38) P2RX7GPR55CNR1CNR2GBA1
SCHEMBL20042743 0.83 P2RX7 (0.40) P2RX7GPR55CNR1CNR2GBA1
SCHEMBL20042674 0.82 P2RX7 (0.37) P2RX7GBA1HSP90AA1KMT2AMEN1
SCHEMBL20042887 0.82 GPR6 (0.42) P2RX7GPR55CNR1CNR2GBA1
SCHEMBL20042836 0.82 P2RX7 (0.43) P2RX7GPR55CNR1CNR2GBA1
SCHEMBL20042872 0.81 P2RX7 (0.44) P2RX7GPR55CNR1CNR2GBA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed