SCHEMBL20042721

SCHEMBL20042721

Cc1nc2c(c(N3CCC3)n1)CN(C(=O)c1cccc(C#N)c1)C2

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 5/20 0.47
P2RX7 Q99572 1/20 0.45
SMO Q99835 1/20 0.42
NAMPT P43490 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
ADORA2A P29274 3/20 0.40
CFTR P13569 1/20 0.40
PRLHR P49683 1/20 0.40
PDE2A O00408 2/20 0.40
MAP3K12 Q12852 1/20 0.39
SLC6A7 Q99884 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042728 0.88 MEN1 (0.42) MEN1KMT2AL3MBTL1PDE2ASLC6A7
SCHEMBL20043028 0.87 KDM4E (0.40) GRM5P2RX7MEN1KMT2AL3MBTL1
SCHEMBL20042668 0.86 HPGD (0.51) GRM5P2RX7MEN1KMT2AL3MBTL1
SCHEMBL20042713 0.85 GRM5 (0.45) GRM5P2RX7MEN1KMT2AL3MBTL1
SCHEMBL20042656 0.85 KDM4E (0.37) GRM5P2RX7MEN1KMT2AL3MBTL1
SCHEMBL20042903 0.85 MEN1 (0.42) P2RX7MEN1KMT2AL3MBTL1CFTR
SCHEMBL20042684 0.85 SMN1; SMN2 (0.52) GRM5P2RX7
SCHEMBL20042771 0.85 P2RX7 (0.47) GRM5P2RX7MEN1KMT2AL3MBTL1
SCHEMBL20042839 0.84 P2RX7 (0.45) P2RX7SMOMEN1KMT2AL3MBTL1
SCHEMBL20042754 0.83 MEN1 (0.41) GRM5P2RX7MEN1KMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed