SCHEMBL20043028

SCHEMBL20043028

Cc1cc(C#N)cc(C(=O)N2Cc3nc(C)nc(N4CCC4)c3C2)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.40
TSHR P16473 4/20 0.40
CASP1 P29466 4/20 0.40
CASP7 P55210 4/20 0.40
HSD17B10 Q99714 4/20 0.40
HPGD P15428 3/20 0.40
KMT2A Q03164 5/20 0.39
MEN1 O00255 4/20 0.39
CFTR P13569 4/20 0.38
ALDH1A1 P00352 5/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
MAPK1 P28482 1/20 0.37
ALOX15 P16050 3/20 0.36
MAPT P10636 2/20 0.36
POLB P06746 2/20 0.36
HTT P42858 1/20 0.36
ALOX12 P18054 1/20 0.36
P2RX7 Q99572 1/20 0.36
TDP1 Q9NUW8 1/20 0.35
GRM5 P41594 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042656 0.90 KDM4E (0.37) KDM4ETSHRCASP1CASP7HSD17B10
SCHEMBL20042713 0.90 GRM5 (0.45) KDM4ETSHRCASP1CASP7HSD17B10
SCHEMBL20042721 0.87 GRM5 (0.47) KMT2AMEN1CFTRL3MBTL1P2RX7
SCHEMBL20042728 0.86 MEN1 (0.42) KMT2AMEN1ALDH1A1L3MBTL1FASN
SCHEMBL20042854 0.84 GRM5 (0.42) KDM4ETSHRCASP1CASP7HSD17B10
SCHEMBL20042743 0.82 P2RX7 (0.40) KDM4ETSHRCASP1CASP7HSD17B10
SCHEMBL20042903 0.82 MEN1 (0.42) KDM4ETSHRCASP1CASP7HSD17B10
SCHEMBL20042707 0.81 P2RX7 (0.40) KDM4ETSHRCASP1CASP7HSD17B10
SCHEMBL20042873 0.81 P2RX7 (0.38) KDM4ETSHRCASP1CASP7HSD17B10
SCHEMBL20042668 0.81 HPGD (0.51) KDM4EHPGDKMT2AMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed