SCHEMBL20042751

SCHEMBL20042751

Cc1nc2c(c(N3CCC3)n1)CN(C(=O)c1ccc(Cl)cc1)C2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.49
GBA1 P04062 4/20 0.46
KMT2A Q03164 2/20 0.45
LMNA P02545 2/20 0.43
POLB P06746 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
USP2 O75604 1/20 0.42
CASP1 P29466 1/20 0.42
CASP7 P55210 1/20 0.42
P2RX7 Q99572 2/20 0.42
MEN1 O00255 1/20 0.41
TACR3 P29371 1/20 0.41
KCNH2 Q12809 1/20 0.41
ALDH1A1 P00352 3/20 0.40
HPGD P15428 3/20 0.40
CHRNA7 P36544 1/20 0.40
PHGDH O43175 1/20 0.40
KDM4E B2RXH2 1/20 0.40
HTT P42858 1/20 0.40
HIF1A Q16665 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042817 0.91 PKM (0.44) GBA1KMT2ALMNAUSP2P2RX7
SCHEMBL20042685 0.88 HTT (0.42) GBA1SMN1; SMN2P2RX7TACR3KCNH2
SCHEMBL20042689 0.88 P2RX7 (0.39) HSD17B10GBA1SMN1; SMN2USP2CASP1
SCHEMBL20042687 0.88 HSD17B10 (0.51) HSD17B10GBA1KMT2ALMNAPOLB
SCHEMBL20042839 0.88 P2RX7 (0.45) GBA1KMT2ASMN1; SMN2P2RX7MEN1
SCHEMBL20042886 0.88 HPGD (0.49) KMT2AP2RX7TACR3HPGD
SCHEMBL20042752 0.88 HPGD (0.47) GBA1KMT2ALMNASMN1; SMN2P2RX7
SCHEMBL20042667 0.87 TACR3 (0.46) P2RX7TACR3KCNH2
SCHEMBL20042811 0.87 HSD17B10 (0.60) HSD17B10GBA1KMT2ALMNAPOLB
SCHEMBL20042771 0.87 P2RX7 (0.47) KMT2ALMNASMN1; SMN2P2RX7MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed