SCHEMBL20042744

SCHEMBL20042744

Cc1nc(O)c2c(n1)CN(C(=O)c1ccccc1)C2

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MTHFD2 P13995 2/20 0.44
P2RX7 Q99572 4/20 0.42
KIF11 P52732 1/20 0.41
HPGD P15428 1/20 0.41
GRM5 P41594 3/20 0.40
ACHE P22303 1/20 0.40
BLM P54132 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
TSHR P16473 1/20 0.39
TRAP1 Q12931 1/20 0.38
KCNH2 Q12809 1/20 0.38
GBA1 P04062 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042734 0.86 P2RX7 (0.47) MTHFD2P2RX7KIF11HPGDGRM5
SCHEMBL20042726 0.85 PKM (0.45) P2RX7GRM5
SCHEMBL20042839 0.81 P2RX7 (0.45) MTHFD2P2RX7HPGDTSHRGBA1
SCHEMBL20042663 0.72 P2RX7 (0.34) P2RX7
SCHEMBL20042685 0.71 HTT (0.42) P2RX7GRM5KCNH2GBA1
SCHEMBL19547099 0.71 P2RX7 (0.42) MTHFD2P2RX7
SCHEMBL20042684 0.70 SMN1; SMN2 (0.52) P2RX7HPGDGRM5TSHRKCNH2
SCHEMBL20042893 0.70 CYP2C19 (0.45) HPGDACHESIGMAR1
SCHEMBL31016562 0.70 C5AR1 (0.39)
SCHEMBL20042817 0.70 PKM (0.44) P2RX7HPGDGBA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed