SCHEMBL20042795

SCHEMBL20042795

O=C(c1ccc(Cl)c(Cl)c1)N1Cc2nc(C3CC3)nc(N3CCC3)c2C1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.46
HTR1A P08908 2/20 0.44
UBE2M P61081 1/20 0.42
DCUN1D1 Q96GG9 1/20 0.42
PKM P14618 1/20 0.41
GPR6 P46095 1/20 0.41
HSD11B1 P28845 1/20 0.40
TSHR P16473 1/20 0.39
PDE10A Q9Y233 2/20 0.39
IDH1 O75874 1/20 0.39
NTSR1 P30989 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042719 0.89 HSD17B10 (0.46) GPR6HSD11B1PDE10ANTSR1
SCHEMBL20042722 0.87 ALDH1A1 (0.43) PKMHSD11B1NTSR1
SCHEMBL20042886 0.84 HPGD (0.49) HPGDHTR1APKMGPR6HSD11B1
SCHEMBL20042725 0.82 PDE2A (0.41) PDE10ANTSR1
SCHEMBL20042752 0.78 HPGD (0.47) HPGDTSHR
SCHEMBL20042887 0.77 GPR6 (0.42) HPGDGPR6TSHR
SCHEMBL20042789 0.77 GPR6 (0.42) HPGDGPR6TSHR
SCHEMBL20042803 0.76 GPR6 (0.40) HPGDGPR6TSHR
SCHEMBL20042792 0.76 TACR3 (0.46) HPGDGPR6
SCHEMBL20042667 0.76 TACR3 (0.46) HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed