SCHEMBL20042863

SCHEMBL20042863

Cc1nc2c(c(N3CCC3)n1)CN(C(=O)c1cc(F)cc(Cl)c1)C2

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 3/20 0.42
KCNH2 Q12809 2/20 0.42
PDE2A O00408 2/20 0.41
P2RX7 Q99572 7/20 0.38
TAS1R3 Q7RTX0 1/20 0.37
TAS1R1 Q7RTX1 1/20 0.37
TAS1R2 Q8TE23 1/20 0.37
TP53 P04637 1/20 0.34
THRB P10828 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
GBA1 P04062 1/20 0.34
NPY5R Q15761 1/20 0.33
PROKR1 Q8TCW9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042829 0.92 P2RX7 (0.41) GRM5KCNH2P2RX7GBA1NPY5R
SCHEMBL20042689 0.92 P2RX7 (0.39) GRM5PDE2AP2RX7TP53THRB
SCHEMBL20042854 0.89 GRM5 (0.42) GRM5P2RX7TP53THRBTDP1
SCHEMBL20042702 0.87 P2RX7 (0.49) P2RX7
SCHEMBL20042656 0.85 KDM4E (0.37) GRM5P2RX7TP53THRBTDP1
SCHEMBL20042725 0.85 PDE2A (0.41) GRM5KCNH2PDE2AP2RX7TAS1R3
SCHEMBL20042713 0.85 GRM5 (0.45) GRM5P2RX7
SCHEMBL20042667 0.84 TACR3 (0.46) KCNH2PDE2AP2RX7
SCHEMBL20042861 0.84 P2RX7 (0.39) GRM5P2RX7
SCHEMBL20042684 0.84 SMN1; SMN2 (0.52) GRM5KCNH2P2RX7TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed