SCHEMBL20042861

SCHEMBL20042861

Cc1nc2c(c(N3CCC3)n1)CN(C(=O)c1cc(Cl)cc(OC(F)(F)F)c1)C2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 5/20 0.39
MGLL Q99685 4/20 0.36
MAPK7 Q13164 1/20 0.34
GPBAR1 Q8TDU6 2/20 0.34
MAPT P10636 1/20 0.33
GRM5 P41594 1/20 0.33
ALDH1A1 P00352 1/20 0.33
DDR1 Q08345 1/20 0.33
KDM4E B2RXH2 1/20 0.32
HPGD P15428 1/20 0.32
TSHR P16473 1/20 0.32
CASP1 P29466 1/20 0.32
CASP7 P55210 1/20 0.32
HSD17B10 Q99714 1/20 0.32
PIK3CD O00329 1/20 0.32
PIK3R1 P27986 1/20 0.32
PIK3CA P42336 1/20 0.32
PIK3CB P42338 1/20 0.32
PIK3CG P48736 1/20 0.32
PIK3R5 Q8WYR1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042707 0.91 P2RX7 (0.40) P2RX7MGLLMAPK7ALDH1A1KDM4E
SCHEMBL20042689 0.87 P2RX7 (0.39) P2RX7MAPTGRM5CASP1CASP7
SCHEMBL20042702 0.86 P2RX7 (0.49) P2RX7MAPTTSHRHSD17B10
SCHEMBL20042705 0.85 EPHX2 (0.45) P2RX7MGLLMAPK7
SCHEMBL20042863 0.84 GRM5 (0.42) P2RX7GRM5
SCHEMBL20042854 0.84 GRM5 (0.42) P2RX7GRM5KDM4EHPGDTSHR
SCHEMBL20042765 0.83 P2RX7 (0.42) P2RX7MGLLMAPK7HPGD
SCHEMBL20042656 0.82 KDM4E (0.37) P2RX7GRM5ALDH1A1KDM4EHPGD
SCHEMBL20042694 0.81 P2RX7 (0.43) P2RX7MGLLMAPK7KDM4EHPGD
SCHEMBL20042780 0.80 P2RX7 (0.43) P2RX7MGLLMAPK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed