SCHEMBL20042829

SCHEMBL20042829

Cc1nc2c(c(N3CCC3)n1)CN(C(=O)c1cc(F)cc(F)c1)C2

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 3/20 0.41
NPY5R Q15761 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.36
GBA1 P04062 4/20 0.34
HTT P42858 1/20 0.34
GRM5 P41594 3/20 0.33
KCNH2 Q12809 2/20 0.33
HPGD P15428 2/20 0.33
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33
GPR55 Q9Y2T6 1/20 0.33
KDM4E B2RXH2 1/20 0.33
TSHR P16473 1/20 0.33
CASP1 P29466 1/20 0.33
CASP7 P55210 1/20 0.33
HSD17B10 Q99714 1/20 0.33
TACR3 P29371 1/20 0.33
MTOR P42345 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042863 0.92 GRM5 (0.42) P2RX7NPY5RGBA1GRM5KCNH2
SCHEMBL20042713 0.90 GRM5 (0.45) P2RX7GRM5HPGDKDM4ETSHR
SCHEMBL20042684 0.89 SMN1; SMN2 (0.52) P2RX7SMN1; SMN2HTTGRM5KCNH2
SCHEMBL20042685 0.88 HTT (0.42) P2RX7SMN1; SMN2GBA1HTTGRM5
SCHEMBL20042743 0.88 P2RX7 (0.40) P2RX7SMN1; SMN2GBA1HPGDCNR1
SCHEMBL20042689 0.86 P2RX7 (0.39) P2RX7SMN1; SMN2GBA1GRM5CNR2
SCHEMBL20042666 0.85 KMT2A (0.46) P2RX7GBA1GRM5KCNH2CNR1
SCHEMBL20042823 0.84 P2RX7 (0.45) P2RX7GBA1HTTHPGDCNR1
SCHEMBL20042836 0.84 P2RX7 (0.43) P2RX7SMN1; SMN2GBA1HTTHPGD
SCHEMBL20042769 0.84 P2RX7 (0.38) P2RX7GBA1CNR1CNR2GPR55

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed