SCHEMBL20042896

SCHEMBL20042896

Cc1nc2c(c(N3CCC3)n1)[C@@H](C)N(C(=O)c1cnc(C)c(Cl)c1)C2

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 10/20 0.38
TACR3 P29371 3/20 0.35
CXCR3 P49682 2/20 0.34
HPGDS O60760 1/20 0.33
P2RY12 Q9H244 1/20 0.33
HCRTR2 O43614 1/20 0.33
LMNA P02545 1/20 0.33
TACR2 P21452 1/20 0.32
TACR1 P25103 1/20 0.32
P2RX7 Q99572 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042766 0.88 TACR3 (0.36) TACR3HCRTR2TACR2TACR1P2RX7
SCHEMBL20042852 0.83 TACR3 (0.47) TACR3TACR2TACR1P2RX7
SCHEMBL20042883 0.83 GPR6 (0.39) TACR3LMNATACR2TACR1P2RX7
SCHEMBL20042983 0.83 GPR6 (0.39) TACR3LMNATACR2TACR1P2RX7
SCHEMBL20042982 0.83 P2RX7 (0.46) TACR3LMNATACR2TACR1P2RX7
SCHEMBL20042851 0.83 P2RX7 (0.46) TACR3LMNATACR2TACR1P2RX7
SCHEMBL20042742 0.82 PROKR1 (0.35) TACR3TACR2P2RX7
SCHEMBL20042868 0.82 P2RX7 (0.35) GRM5TACR3LMNATACR2TACR1
SCHEMBL20042727 0.82 TACR3 (0.47) TACR3TACR2TACR1P2RX7
SCHEMBL20042878 0.82 TACR3 (0.47) TACR3TACR2TACR1P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed