SCHEMBL2004407

SCHEMBL2004407

O=C(c1noc(-c2ccccn2)n1)c1c(C(F)(F)F)n(Cc2ccc(Cl)cc2)c2ccccc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.40
CES1 P23141 1/20 0.40
MCL1 Q07820 3/20 0.37
S1PR1 P21453 1/20 0.37
S1PR3 Q99500 1/20 0.37
STAT3 P40763 2/20 0.36
CTSD P07339 1/20 0.36
GUSB P08236 1/20 0.36
PTGES2 Q9H7Z7 1/20 0.36
ALDH1A1 P00352 2/20 0.35
POLB P06746 2/20 0.35
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
USP2 O75604 1/20 0.35
LMNA P02545 1/20 0.35
KMT2A Q03164 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2005678 0.91 STAT3 (0.35) STAT3PTGES2ALDH1A1POLBKDM4E
SCHEMBL2002093 0.90 LMNA (0.40) FAAHCES1ALDH1A1POLBMEN1
SCHEMBL2006169 0.88 FAAH (0.43) FAAHCES1MCL1CTSDGUSB
SCHEMBL2006154 0.87 DRD2 (0.37) S1PR3STAT3PTGES2ALDH1A1POLB
SCHEMBL2003713 0.86 MCL1 (0.39) MCL1CTSDGUSBPTGES2ALDH1A1
SCHEMBL2004941 0.85 GRM5 (0.38) FAAHCES1ALDH1A1MEN1LMNA
SCHEMBL2001534 0.85 HDAC6 (0.41) S1PR1PTGES2ALDH1A1POLBKDM4E
SCHEMBL2005704 0.83 FAAH (0.39) FAAHCES1MCL1PTGES2ALDH1A1
SCHEMBL2002391 0.82 L3MBTL1 (0.39) FAAHCES1S1PR3ALDH1A1MEN1
SCHEMBL2004742 0.82 STAT3 (0.35) FAAHSTAT3PTGES2ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed