SCHEMBL2005502

SCHEMBL2005502

O=C(c1noc(-c2ccncn2)n1)c1c(C(F)(F)F)n(Cc2ccc(Cl)cc2Cl)c2ccccc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.38
MAPT P10636 2/20 0.38
ALDH1A1 P00352 1/20 0.38
ALOX12 P18054 1/20 0.38
CYP1A2 P05177 2/20 0.36
CYP2D6 P10635 2/20 0.36
CYP2C9 P11712 2/20 0.36
NPSR1 Q6W5P4 2/20 0.36
CYP3A4 P08684 1/20 0.36
TSHR P16473 1/20 0.36
PMP22 Q01453 1/20 0.36
HIF1A Q16665 1/20 0.36
VDR P11473 1/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
CYP2C19 P33261 1/20 0.35
MAPK14 Q16539 3/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
TP53 P04637 1/20 0.33
SCD O00767 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2005893 0.94 SCD (0.34) LMNAMAPTALDH1A1ALOX12CYP1A2
SCHEMBL2002093 0.91 LMNA (0.40) LMNAMAPTALDH1A1ALOX12CYP1A2
SCHEMBL2005962 0.91 L3MBTL1 (0.35) LMNAMAPTALDH1A1ALOX12MAPK14
SCHEMBL2005678 0.91 STAT3 (0.35) LMNAMAPTALDH1A1CYP1A2CYP2D6
SCHEMBL2009499 0.90 FAAH (0.33) LMNAMAPTALDH1A1ALOX12CYP1A2
SCHEMBL2008605 0.90 LMNA (0.41) LMNAMAPTALDH1A1ALOX12CYP1A2
SCHEMBL2012645 0.89 LMNA (0.40) LMNAMAPTALDH1A1ALOX12CYP1A2
SCHEMBL2002685 0.88 PLA2G2A (0.37) LMNAMAPTALDH1A1CYP1A2CYP2D6
SCHEMBL2004879 0.88 ALOX5AP (0.33) LMNAMAPTCYP2C9CYP3A4SMN1; SMN2
SCHEMBL2007450 0.87 LMNA (0.38) LMNAMAPTALDH1A1ALOX12CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed