SCHEMBL2004879

SCHEMBL2004879

CCOc1ccc2c(c1)c(C(=O)c1noc(-c3ccncn3)n1)c(C(F)(F)F)n2Cc1ccc(Cl)cc1Cl

nearest known ligand 0.33

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 3/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
F2RL3 Q96RI0 1/20 0.32
LMNA P02545 2/20 0.32
MAPT P10636 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
ALOX5 P09917 1/20 0.32
SLC26A4 O43511 1/20 0.32
POLB P06746 1/20 0.32
SCD O00767 1/20 0.31
SCD5 Q86SK9 1/20 0.31
EIF4EBP1 Q13541 1/20 0.31
PLA2G2A P14555 1/20 0.30
STAT3 P40763 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2002685 0.94 PLA2G2A (0.37) ALOX5APCYP3A4CYP2C9F2RL3LMNA
SCHEMBL2005091 0.92 ALOX5AP (0.39) ALOX5APALOX5STAT3
SCHEMBL2005893 0.92 SCD (0.34) CYP3A4CYP2C9LMNAMAPTSCD
SCHEMBL2003268 0.91 ALOX5AP (0.36) ALOX5APCYP3A4CYP2C9F2RL3LMNA
SCHEMBL2003150 0.91 S1PR1 (0.35) ALOX5APCYP3A4CYP2C9F2RL3LMNA
SCHEMBL2002148 0.91 LMNA (0.34) ALOX5APCYP3A4CYP2C9LMNAMAPT
SCHEMBL2009499 0.90 FAAH (0.33) CYP3A4CYP2C9LMNAMAPTSMN1; SMN2
SCHEMBL2005962 0.89 L3MBTL1 (0.35) LMNAMAPTSCDSCD5
SCHEMBL2002732 0.88 LMNA (0.33) ALOX5APCYP3A4CYP2C9F2RL3LMNA
SCHEMBL2005502 0.88 LMNA (0.38) CYP3A4CYP2C9LMNAMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed