SCHEMBL2009499

SCHEMBL2009499

Cc1ccc2c(c1)c(C(=O)c1noc(-c3ccncn3)n1)c(C(F)(F)F)n2Cc1ccc(Cl)cc1Cl

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.33
MAPK14 Q16539 3/20 0.33
SCD O00767 1/20 0.32
SCD5 Q86SK9 1/20 0.32
MAPK1 P28482 2/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
KDM4E B2RXH2 1/20 0.32
PTGS1 P23219 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.32
MALT1 Q9UDY8 1/20 0.31
CYP2C9 P11712 2/20 0.31
CYP3A4 P08684 1/20 0.31
EIF4EBP1 Q13541 1/20 0.31
LMNA P02545 2/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
TP53 P04637 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2005893 0.95 SCD (0.34) MAPK14SCDSCD5MAPK1MEN1
SCHEMBL2005962 0.92 L3MBTL1 (0.35) MAPK14SCDSCD5MAPK1LMNA
SCHEMBL1999358 0.92 FAAH (0.41) FAAHMAPK14SCDSCD5MEN1
SCHEMBL2002685 0.91 PLA2G2A (0.37) MAPK1MEN1KMT2APTGDR2CYP2C9
SCHEMBL2006492 0.90 GRM5 (0.35) FAAHMEN1KMT2ACYP2C9CYP3A4
SCHEMBL2005502 0.90 LMNA (0.38) MAPK14SCDSCD5MEN1KMT2A
SCHEMBL2001504 0.90 FAAH (0.35) FAAHMAPK14MAPK1MEN1KMT2A
SCHEMBL2004879 0.90 ALOX5AP (0.33) SCDSCD5CYP2C9CYP3A4EIF4EBP1
SCHEMBL2008461 0.89 RET (0.36) FAAHMAPK1MEN1KMT2AKDM4E
SCHEMBL2005516 0.88 FAAH (0.33) FAAHMAPK14SCDSCD5MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed