SCHEMBL2005563

SCHEMBL2005563

O=C(c1cnc(-c2ccccc2)o1)c1c(Cl)n(Cc2ccc(Cl)cc2Cl)c2ccccc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.45
MAPT P10636 3/20 0.45
CYP1A2 P05177 2/20 0.45
CYP2D6 P10635 2/20 0.45
CYP2C9 P11712 2/20 0.45
NPSR1 Q6W5P4 2/20 0.45
ALDH1A1 P00352 2/20 0.45
ALOX12 P18054 1/20 0.45
CYP3A4 P08684 1/20 0.45
TSHR P16473 1/20 0.45
PMP22 Q01453 1/20 0.45
HIF1A Q16665 1/20 0.45
VDR P11473 1/20 0.39
CCR2 P41597 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
TP53 P04637 2/20 0.39
SLC9A1 P19634 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1999686 0.95 MAPT (0.42) LMNAMAPTCYP1A2CYP2D6CYP2C9
SCHEMBL2006426 0.94 LMNA (0.43) LMNAMAPTCYP1A2CYP2D6CYP2C9
SCHEMBL2008737 0.92 LMNA (0.42) LMNAMAPTCYP1A2CYP2D6CYP2C9
SCHEMBL2008306 0.92 L3MBTL1 (0.43) LMNAMAPTCYP1A2CYP2D6CYP2C9
SCHEMBL2008233 0.91 LMNA (0.39) LMNAMAPTCYP1A2CYP2D6CYP2C9
SCHEMBL2002616 0.89 ALDH1A1 (0.45) LMNAMAPTCYP1A2CYP2D6CYP2C9
SCHEMBL2002932 0.89 PLA2G2A (0.43) LMNAMAPTCYP1A2CYP2C9ALDH1A1
SCHEMBL1996469 0.88 LMNA (0.42) LMNAMAPTCYP1A2CYP2D6CYP2C9
SCHEMBL2011328 0.88 LMNA (0.40) LMNAMAPTCYP1A2CYP2D6CYP2C9
SCHEMBL2004385 0.88 LMNA (0.43) LMNAMAPTCYP1A2CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed