SCHEMBL2005616

SCHEMBL2005616

COc1ccc2c(c1)c(C(=O)c1nc3ncccc3o1)c(C)n2Cc1ccc(Cl)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.51
TSHR P16473 3/20 0.51
PKM P14618 2/20 0.51
MAPT P10636 2/20 0.51
MEN1 O00255 1/20 0.51
RGS12 O14924 1/20 0.51
LMNA P02545 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2C9 P11712 1/20 0.51
NFKB1 P19838 1/20 0.51
MAPK1 P28482 1/20 0.51
CYP2C19 P33261 1/20 0.51
GNAI1 P63096 1/20 0.51
PMP22 Q01453 1/20 0.51
KMT2A Q03164 1/20 0.51
HIF1A Q16665 1/20 0.51
PLA2G2A P14555 7/20 0.49
FAAH O00519 2/20 0.45
HTT P42858 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1999688 0.88 PTGDR2 (0.43) ALDH1A1TSHRPKMMAPTMEN1
SCHEMBL3007027 0.87 PLA2G2A (0.53) ALDH1A1TSHRPKMMAPTMEN1
SCHEMBL3002846 0.85 FAAH (0.55) ALDH1A1TSHRPKMMAPTMEN1
SCHEMBL2003055 0.83 ALDH1A1 (0.52) ALDH1A1TSHRPKMMAPTMEN1
SCHEMBL2005823 0.83 ALDH1A1 (0.52) ALDH1A1TSHRPKMMAPTMEN1
SCHEMBL12628702 0.82 LMNA (0.49) ALDH1A1MAPTLMNAPLA2G2AFAAH
SCHEMBL2999029 0.82 MEN1 (0.49) ALDH1A1TSHRPKMMAPTMEN1
SCHEMBL2002995 0.82 ALDH1A1 (0.55) ALDH1A1TSHRPKMMAPTMEN1
SCHEMBL2006827 0.82 ALDH1A1 (0.56) ALDH1A1TSHRPKMMAPTMEN1
SCHEMBL12629109 0.81 PTGS2 (0.42) MEN1KMT2APTGS2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed